Ki value nM Dopamine D2 receptor | Daily Defined Dose (DDD) | Chlorpromazine Equivalent Ratio (EQ) | |
---|---|---|---|
Loose binding or partial agonism | |||
Quetiapinea | 122 | 400 mg | 0.80 |
Clozapinea | 63 | 300 mg | 1.50 |
Cariprazinec | 18.0 | 3 mg | 100 |
Olanzapinea | 5.1 | 10 mg | 30 |
Amisulprideb | 1.8 | 400 mg | 0.86 |
Aripiprazoleb | 1.8 | 15 mg | 20.0 |
Tight binding | |||
Dopaminea | 1.75 | - | - |
Lurasidonec | 1.68 | 60 mg | 16 |
Paliperidoneb | 1.6 | 6 mg/2.5 mg | 66.7 |
Risperidonea | 1.1 | 5 mg/1.8 mg | 100 |
Haloperidola | 0.55 | 8 mg | 60.0 |
Zuclopenthixold | Comparable to Haloperidol | 30 mg/15 mg | 12 |